Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_04452
Ion Channel
Voltage-gated potassium channel subfamily H member 2
Peptide Function
Blocker
Gene Name
KCNH2
Activity Data (nM)
IC50
Not available
Ki
Not available
EC50
Not available
Kd
9.9 nM
Biologically Active
Not specified
Sequence Information
Peptide Sequence
DRDSCVDKSRCAKYGYYQECQDCCKNAGHNGGTCMFFKCKCA
Peptide UniProt Accession
UniParc
UPI000007DD22
Peptide Synonyms/Alias
CeErg4
Peptide Species
Centruroides elegans (Bark scorpion)
Peptide Name
Potassium channel toxin gamma-KTx 1.7
CAS Number
Not available
Experimental Conditions
pH
pH 7.2
Holding Potential (mV)
−70 mV
Temperature
21–23 °C
Test Method
Patch-clamping
Test Species
CHO cell (Chinese hamster ovary cell)
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
VGKCs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)
References & Disease Information
Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available